Drugs.com provides accurate and independent information on more than 24,000 prescription drugs, over-the-counter medicines and natural products. (14)C-Labeled ethylenediamine (EDA) was accumulated by slices of adult rat cerebral cortex, although the tissue:medium ratios were much lower than those for gamma-aminobutyric acid.EDA uptake was temp-dependent and appeared to take place by both sodium dependent and sodium independent mechanisms. This means it is still under development and may contain inaccuracies. The biochemical and antioxidant properties of chitosan modified with acetylacetone and ethylenediamine (Cacen) or diethylenetriamine (Cacdien) associated with ceftazidime (F) were investi … Biological properties of chitosan derivatives associated with the ceftazidime drug Carbohydr Polym. Phenolic ethylenediamine derivatives: a study of orally effective iron chelators. Inhibition studies indicate that ethylenediamine may be transported in part by the small … ethanolamine derivatives; ethylenediamine derivatives; first gen. antihist. Ethylenediamine derivatives possessing a substituent at the C1 position in S configuration and phenylenediamine derivatives possessing a substituent at the C5 position demonstrated moderate to strong anti-fXa activity. b) Ethylenediamine derivatives. Other uses antihistamine drugs. Identification Name Ethylenediamine Accession Number DB14189 Description. This formulary is subject to change throughout the year and plan exclusions may override this list. Drug Drug Description; Tripelennamine: A histamine H1 antagonist used to treat hypersensitivity reactions, coughs, and the common cold. ethylenediamine derivatives heterocycle aromatic ring compounds general formula Prior art date 2000-04-05 Application number PCT/JP2001/002945 Other languages French (fr) Japanese (ja) Inventor Toshiharu Yoshino Tsutomu Nagata Noriyasu Haginoya Kenji Yoshikawa Hideyuki Kanno Masatoshi Nagamochi Original Assignee Daiichi Pharmaceutical Co., Ltd. Result indicated that the ethylenediamine derivatives, N,N-Bis(2-hydroxy-5-bromobenzyl)-1,2- ethanediamine (21), and N,N-Bis(2-hydroxy-5-chlorobenzyl)-1,2-ethanediamine (22) showed the most favorable antimicrobial activity exhibiting LC50 of 11.6 and 8.79 μM against S.enterica, 86 and 138 μM against P. aeruginosa, and 140 and 287 μM against S. aureus, respectively. Ethylenediamine Derivatives. We designed an amino acid type PEG (aaPEG) for preparation of a multi- 1999 Mar;73(3):145-9. doi: 10.1016/s0162-0134(99)00009-4. Precursor to chelation agents, drugs, and agrochemicals A most prominent derivative of ethylenediamine is the chelating agent EDTA, which is derived from ethylenediamine via a Strecker synthesis involving cyanide and formaldehyde. Ethambutol is an ethylenediamine derivative that is ethane-1,2-diamine in which one hydrogen attached to each of the nitrogens is sutstituted by a 1-hydroxybutan-2-yl group (S,S-configuration). Data sources include IBM Watson Micromedex (updated 6 Jan 2021), Cerner Multum™ (updated 4 Jan 2021), ASHP … ChEBI Name ethambutol: ChEBI ID CHEBI:4877: Definition An ethylenediamine derivative that is ethane-1,2-diamine in which one hydrogen attached to each of the nitrogens is sutstituted by a 1-hydroxybutan-2-yl group (S,S-configuration).It is a bacteriostatic antimycobacterial drug, effective against Mycobacterium tuberculosis and some other mycobacteria. Results and discussion 2.1. • These are clinically used in the treatment of histamine mediated allergic conditions like allergic rhinitis, allergic conjuctivitis etc., CLASSIFICATION: a) Amino alkyl ethers. It is scheduled to be annotated soon. Ethylenediamine is an organic compound that is used as a building block for the production of many other chemical products. View more via ChEBI Ontology . 3. ChemInform Abstract: ULTRA-SHORT-ACTING β-ADRENERGIC RECEPTOR BLOCKING AGENTS. February 2012; Medicinal chemistry (Shāriqah (United Arab Emirates)) 8(2):252-65 derivatives, misc. Benefit designs may vary with respect to drug coverage, quantity limits, days supply and prior authorization. Name Ethylenediamine Derivatives Accession Number DBCAT003721 Description Not Available Drugs. Biochemical, morphochemical and pharmacodynamic evaluation of accumulation of ethylenediamine derivatives (ROM-203, MK-142) in some rat tissues Mater Med Pol. PLEASE NOTE: Because prescription drug programs vary by group, the inclusion of a drug in this formulary does not imply coverage. 2019 Oct 15;222:115002. doi: 10.1016/j.carbpol.2019.115002. General pharmacological properties. Poly(amidoamine), or PAMAM, is a class of dendrimer which is made of repetitively branched subunits of amide and amine functionality.PAMAM dendrimers, sometimes referred to by the trade name Starburst, have been extensively studied since their synthesis in 1985, and represent the most well-characterized dendrimer family as well as the first to be commercialized. Usually, PEG is converted to a carboxyl derivative and conju-gated with a protein as a simple acyl moiety. [Pharmacological study of new ethylenediamine derivatives with antiarrhythmic activity]. Jul-Sep 1977;9(3):216-24. Title:2D Chemometrics Analyses of Tetrahydroquinoline and Ethylenediamine Derivatives with Antimalarial Activity VOLUME: 8 ISSUE: 2 Author(s): Humberto Fonseca de Freitas and Marcelo Santos Castilho Affiliation:Faculdade de Farmacia, Universidade Federal da Bahia (UFBA), Salvador, Bahia, 40170-115. development of novel drug-carrier systems, although its sim-ple structure limits the types of hybrids that can be produced. ethylenediamine: ChEBI ID CHEBI:30347: Definition An alkane-α,ω-diamine in which the alkane is ethane. Compounds of the general formula (1): Q1-Q2-C(=O)-N(R?1)-Q3-N(R2)-T1-Q4¿; and drugs which contain the compounds and are efficacious for thrombosis and embolism. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.) Ethylenediamine-palladium(II) complexes with pyridine and its derivatives: synthesis, molecular structure and initial antitumor studies J Inorg Biochem .
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